Цымбал С.А. The Copper Reduction Potential Determines the Reductive Cytotoxicity: Relevance to the Design of Metal–Organic Antitumor Drugs. MDPI. 2024. Vol. 29. No. 5. pp. 1032.
Rusina P., Lisov A., Denisova A., Gandalipov E.R., Novikov F., Shtil A.A. Clinical CDK2 Inhibitors: Trends to Selectivity and Efficacy. Recent Patents on Anti-cancer Drug Discovery. 2023. Vol. 18. No. 2. pp. 102-107.
Guk D., Gibadullina K.R., Burlutskiy R.O., Pavlov K.G., Moiseeva A., Tafeenko V.A., Lyssenko K.A., Gandalipov E.R., Shtil A., Beloglazkina E. New Titanocene (IV) Dicarboxylates with Potential Cytotoxicity: Synthesis, Structure, Stability and Electrochemistry. International Journal of Molecular Sciences. 2023. Vol. 24. No. 4. pp. 3340.
Kokinos E.K., Tsymbal S.A., Galochkina A.V., Bezlepkina S.A., Nikolaeva J.V., Vershinina S.O., Shtro A., Tatarskiy V.V., Shtil A.A., Broude E.V., Roninson I.B., Dukhinova M. Inhibition of Cyclin-Dependent Kinases 8/19 Restricts Bacterial and Virus-Induced Inflammatory Responses in Monocytes. Viruses. 2023. Vol. 15. No. 6. pp. 1292.
Kuchur O.A., Zavisrskiy A.V., Shtil А. Transcriptional Reprogramming Regulates Tumor Cell Survival in Response to Ionizing Radiation: a Role of p53. Bulletin of Experimental Biology and Medicine. 2023. Vol. 174. No. 5. pp. 659-665.
Моделирование резистентности хронического миелоидного лейкоза к ингибиторам BCR-ABL в костном мозге
СИНТЕТИЧЕСКАЯ ЛЕТАЛЬНОСТЬ КЛЕТОК MYCN ПОЛОЖИТЕЛЬНОЙ НЕЙРОБЛАСТОМЫ ПОД ДЕЙСТВИЕМ СЕЛЕКТИВНЫХ ИНГИБИТОРОВ CDK2
Цымбал С.А., Штиль А.А. Исследование переносимости медьсодержащих соединений и восстановителя для разработки модели терапии опухолевого асцита. Вопросы онкологии [Voprosy Onkologii]. 2022. Т. 68. № S3. С. 361-362.
Определение цитотоксической и противоопухолевой активности комбинации медьорганических соединений и N-ацетилцистеина на модели полостных метастазов in vivo
Механизмы гибели опухолевых клеток при действии производных териндолона
Кокинос Е.К., Кузьмина Д., Кучур О.А., Цымбал С.А., Василичин В.А., Галочкина А.В., Завирский А.В., Башарин В.А., Штро А.А., Штиль А.А., Духинова М.С. Фенотипический и функциональный анализ линии моноцитов THP-1 как модели воспаления [Phenotypic and functional characteristic analysis of THP-1 cell line as a model of inflammation]. Иммунология [Immunologiya]. 2022. Т. 43. № 3. С. 277-287.
Ivanov V., Agamennone M., Iusupov I.R., Laghezza A., Novoselov A.M., Manasova E.V., Altieri A., Tortorella P., Shtil А., Kurkin A.V. Het(aryl)isatin to het(aryl)aminoindoline scaffold hopping: A route to selective inhibitors of matrix metalloproteinases. Arabian Journal of Chemistry. 2022. Vol. 15. No. 1. pp. 103492.
Ингибирование СDK8/19-зависимого перепрограммирования транскрипции - новый механизм радиосенситизации p53-положительных опухолевых клеток
Shutkov I., Okulova Y.N., Tyurin V.Y., Sokolova E.V., Babkov D.A., Spasov A.A., Gracheva Y.A., Schmidt G., Kirsanov K., Shtil А., Redkozubova O., Shevtsova E.F., Milaeva E.R., Ott I., Nazarov A.A. Ru (III) Complexes with lonidamine-modified ligands. International Journal of Molecular Sciences. 2021. Vol. 22. No. 24. pp. 13468.
Использование меди N-ацетилцистеином и аскорбатом для преодоления лекарственной устойчивости опухолевых клеток
Tsymbal S., Agadzhanyan N., Shtil А. Oxidative stress associated with Cu2+to Cu+ reduction for eradicating wild type and multidrug-resistant tumor cells. Annals of Oncology. 2021. Vol. 32. No. Suppl.6. pp. S1365-S1365.
Kuchur O.A., Kuchur P.D., Kuzmina D., Zavirsky A.V., Shtil A. Differential Regulation of BBC3/PUMA and PMAIP1/Noxa in Ionizing Radiation: the Role of p53. Cell and Tissue Biology. 2021. Vol. 15. No. 6. pp. 544-553.
Bruter А., Rodionova M., Varlamova Е., Shtil А. Super-Enhancers in the Regulation of Gene Transcription: General Aspects and Antitumor Targets. Acta Naturae (англоязычная версия). 2021. Vol. 13. No. 1. pp. 4-15.
Kuchur O.A., Kuzmina D., Dukhinova M.S., Shtil A. The p53 Protein Family in the Response of Tumor Cells to Ionizing Radiation: Problem Development. Acta Naturae (англоязычная версия). 2021. Vol. 13. No. 3. pp. 65-76.
Кучур О.А., Кучур П.Д., Кузьмина Д.О., Завирский А.В., Штиль А.А. Дифференциальная регуляция BBC3/PUMA и PMAIP1/Noxa при ионизирующем излучении: роль p53 [Differential Regulation of BBC3/PUMA and PMAIP1/Noxa by Ionizing Radiation: A Role for p53]. Цитология [Tsitologiya]. 2021. Т. 63. № 4. С. 363-372.
Kuchur O.A., Zavirskiy A.V., Shtil А. Attenuation of p53 signaling by CDK8/19 sensitizes tumor cells to ionizing radiation. Annals of Oncology. 2021. Vol. 32. No. Suppl.6. pp. S1358-S1358.
Tsymbal S.A., Moiseeva A., Agadzhanian N., Efimova S., Markova A.A., Guk D., Krasnovskaya O., Alpatova V., Zaitsev A.V., Shibaeva A., Tatarskiy V.V., Dukhinova M.S., Ol’Shevskaya V., Ostroumova O., Beloglazkina E., Shtil А. Copper-Containing Nanoparticles and Organic Complexes: Metal Reduction Triggers Rapid Cell Death via Oxidative Burst. International Journal of Molecular Sciences. 2021. Vol. 22. No. 20. pp. 11065.
65P - Oxidative stress associated with Cu2+ to Cu+ reduction for eradicating wild type and multidrug resistant tumor cells
Кучур О.А., Кузьмина Д.О., Духинова М.С., Штиль А.А. Белки семейства p53 в ответе опухолевых клеток на ионизирующее излучение: развитие проблемы. Acta Naturae (русскоязычная версия). 2021. Т. 13. № 3. С. 65-76.
Брутер А.В., Родионова М.Д., Варламова Е.А., Штиль А.А. Суперэнхансеры в регуляции транскрипции генов: общебиологические аспекты и мишени противоопухолевой терапии. Acta Naturae (русскоязычная версия). 2021. Т. 13. № 1. С. 4-15.
Механизмы усиления гибели опухолевых клеток при ионизирующем излучении: связь между p53 и CDK8/19
ИНГИБИРОВАНИЕ p53 ЧЕРЕЗ CDK8/19 ПОВЫШАЕТ ЧУВСТВИТЕЛЬНОСТЬ ОПУХОЛЕВЫХ КЛЕТОК К ИОНИЗИРУЮЩЕМУ ИЗЛУЧЕНИЮ
Attenuation of p53 signaling by CDK8/19 sensitizes tumor cells to ionizing radiation
Medvedeva G., Kuzmina D., Nuzhina J.V., Shtil A.A., Dukhinova M.S. How macrophages become transcriptionally dysregulated: A hidden impact of antitumor therapy. International Journal of Molecular Sciences. 2021. Vol. 22. No. 5. pp. 2662.
РОЛЬ СТАТУСА Р53 В ОТВЕТЕ ОПУХОЛЕВЫХ КЛЕТОК НА ИОНИЗИРУЮЩЕЕ ИЗЛУЧЕНИЕ ПРИ ИНГИБИРОВАНИИ CDK8/19
Single vs Multiple Drug Targets: Revising the Therapeutic Concept to Combat Intractable Cancers
Boron-Based Compounds: Potential and Emerging Applications in Medicine
Молекулярные механизмы чувствительности опухолевых клеток к терапевтическому ионизирующему излучению: p53 и CDK8/19
PHOTOCURABLE FILMS BASED ON FIBROIN AND GELATIN FOR REGENERATION OF SKIN COVER
Комбинированное применение наночастиц оксида меди и N-ацетилцистеина для преодоления лекарственной устойчивости опухолевых клеток
The role of p53 status in response to ionizing radiation
Belousov A.V., Morozov V.N., Krusanov G.A., Moiseev A.N., Davydov A.S., Shtil A.A., Klimanov V.A., Kolyvanova M.A., Samoylov A.S. The Change in the Linear Energy Transfer of a Clinical Proton Beam in the Presence of Gold Nanoparticles. Biophysics. 2020. Vol. 65. No. 4. pp. 541-547.
Morozov K.V., Kolyvanova M.A., Kartseva M.E., Shishmakova E.M., Dement’Eva O.V., Isagulieva A.K., Salpagarov M.H., Belousov A.V., Rudoy V.M., Shtil A.A., Samoylov A.S., Morozov V.N. Radiosensitization by gold nanoparticles: impact of the size, dose rate, and photon energy. Nanomaterials. 2020. Vol. 10. No. 5. pp. 952.
Markova A.A., Belyaeva E.V., Radchenko A.S., Dmitrieva M.V., Sigan A.L., Shtil A.A., Chkanikov N.D. Perfluorocarbon nanoemulsions containing fluorinated photosensitizer for photodynamic cancer therapy. IOP Conference Series: Materials Science and Engineering. 2020. Vol. 848. No. 1. pp. 012054.
Morozov V.N., Belousov A.V., Zverev V.I., Shtil A.A., Kolyvanova M.A., Krivoshapkin P.V. The Prospects of Metal Oxide Nanoradiosensitizers: The Effect of the Elemental Composition of Particles and Characteristics of Radiation Sources on Enhancement of the Adsorbed Dose. Biophysics. 2020. Vol. 65. No. 4. pp. 533-540.
Kostyukov A.A., Egorov A.E., Mestergazi M.G., Shmykova A.M., Podrugina T.A., Borissevitch I.E., Shtil A.A., Kuzmin V.A. Photochemical properties of new bis-cyanine dye as a promising agent for in vivo imaging. Mendeleev Communications. 2020. Vol. 30. No. 4. pp. 442-444.
Gornostaev L.M., Fominykh O.I., Rukovets T.A., Lavrikova T.I., Khalyavina J.G., Shtil A.A., Shunaev A.V., Dunaev S.F., Murashova E.V., Chernyshev V.V. Synthesis of 6b, 11b-dihydroxy-12-methylphenyl-11b, 12-dihydrobenzo-[g] indeno [1, 2-b] indole-5, 6, 7 (6b H)-triones and 2-(3-hydroxy-4, 9-dioxo-4, 9-dihydro-1 H-benzo [f] indol-2-yl) benzamides, their structure and antiproliferative activity. Chemistry of Heterocyclic Compounds. 2020. Vol. 56. No. 1. pp. 47-54.
Gornostaev L.M., Fominykh O.I., Rukovets T.A., Lavrikova T.I., Khalyavina J.G., Shtil A., Shunaev A.V., Dunaev S.F., Murashova E.V., Chernyshev V.V. Synthesis of 6b,11b-dihydroxy-12-methylphenyl-11b,12-dihydrobenzo- [g]indeno[1,2-b]indole-5,6,7(6bH)-triones and 2-(3-hydroxy-4,9-dioxo-4,9-dihydro-1H-benzo[f]indol-2-yl)benzamides, their structure and antiproliferative activity. Chemistry of Heterocyclic Compounds. 2020. Vol. 56. No. 1. pp. 47-54.
Silaeva Y.Y., Kalmykov V.A., Varlamova E.A., Korshunov E.N., Korshunova D.S., Kubekina M.V., Shtil A.A., Roninson I.B., Deykin A.V. Genome editing as an approach to the study of in vivo transcription reprogramming. Doklady Biochemistry and Biophysics. 2020. Vol. 490. No. 1. pp. 43-46.
Kotliarova M.S., Soldatenko A.S., Arkhipova A.Y., Bessonov I.V., Davydova L.I., Moysenovich A.M., Bogush V.G., Debabov V.G., Shtil A.A., Moisenovich M.M., Shaitan K.V. Photocurable Films Based on Fibroin and Gelatin for Skin Regeneration. Moscow University Biological Sciences Bulletin. 2020. Vol. 75. No. 1. pp. 20-25.
Beniaminov A.D., Chashchina G.V., Livshits M.A., Kechko O.I., Mitkevich V.A., Mamaeva O.K., Tevyashova A.N., Shtil A.A., Shchyolkina A.K., Kaluzhny D.N. Discrimination between G/C Binding Sites by Olivomycin A Is Determined by Kinetics of the Drug-DNA Interaction. International Journal of Molecular Sciences. 2020. Vol. 21. No. 15. pp. 5299.
Kuchur O.A., Tsymbal S.A., Shestovskaya M.V., Serov N.S., Dukhinova M.S., Shtil A.A. Metal-derived nanoparticles in tumor theranostics: Potential and limitations. Journal of Inorganic Biochemistry. 2020. Vol. 209. pp. 111117.
Marsova M., Odorskaya M., Novichkova M., Polyakova V., Abilev S., Kalinina E., Shtil A., Poluektova E., Danilenko V. The Lactobacillus brevis 47 f strain protects the murine intestine from enteropathy induced by 5-fluorouracil. Microorganisms. 2020. Vol. 8. No. 6. pp. 876.
Bessonov I., Moysenovich A., Arkhipova A., Ezernitskaya M., Efremov Y., Solodilov V., Timashev P., Shaytan K., Shtil A., Moisenovich M. The mechanical properties, secondary structure, and osteogenic activity of photopolymerized fibroin. Polymers. 2020. Vol. 12. No. 3. pp. 646.
Dukhinova M.S., Shestovskaya M.V., Shtil A.A. Metal Nanoparticles in Immunotherapy: Applications, Limitations and Pespectives. Research & Development in Material Science. 2020. Vol. 12(4). No. 3. pp. 1292-1295.
Vasilichin V.A., Tsymbal S.A., Fakhardo A.F., Anastasova E., Marchenko A.S., Shtil A., Vinogradov V.V., Koshel E. Effects of Metal Oxide Nanoparticles on Toll-Like Receptor mRNAs in Human Monocytes. Nanomaterials. 2020. Vol. 10. No. 1. pp. 127.
Moysenovich A.M., Moisenovich M.M., Sudina A.K., Tatarskiy V., Khamidullina A.I., Yastrebova M.A., Davydova L.I., Bogush V.G., Debabov V.G., Arkhipova A.Y., Shaitan K.V., Shtil A.A., Demina I.A. Recombinant Spidroin Films Attenuate Individual Markers of Glucose Induced Aging in NIH 3T3 Fibroblasts. Biochemistry (Moscow). 2020. Vol. 85. No. 7. pp. 808–819.
Tikhomirov A.S., Litvinova V., Andreeva D.V., Tsvetkov V., Dezhenkova L.G., Volodina Y.L., Kaluzhny D.N., Treshalin I., Schols D., Ramonova A.A., Moisenovich M.M., Shtil A.A., Shchekotikhin A.E. Amides of pyrrole- and thiophene-fused anthraquinone derivatives: A role of the heterocyclic core in antitumor properties. European Journal of Medicinal Chemistry. 2020. Vol. 199. pp. 112294.
Moysenovich A.M., Tatarskiy V.V., Yastrebova M.A., Bessonov I.V., Arkhipova A.Y., Kolosov A.S., Davydova L.I., Khamidullina A.I., Bogush V.G., Debabov V.G., Shaitan K.V., Shtil A.A., Moisenovich M.M. Akt and Src mediate the photocrosslinked fibroin-induced neural differentiation. NeuroReport. 2020. Vol. 31. No. 10. pp. 770–775.
Vasilyeva S.V., Petrova A.S., Shtil A.A., Stetsenko D.A. Application of silicon dioxide nanoparticles modified with tumor-targeting ligands for cellular delivery of nucleoside triphosphate analogues. Journal of Saudi Chemical Society. 2020. Vol. 24. No. 1. pp. 98-104.
Sagnou M., Novikov F.N., Ivanova E.S., Alexiou P., Stroylov V.S., Titov I.Y., Tatarskiy V., Vagida M.S., Pelecanou M., Shtil A.A., Chilov G.G. Novel curcumin derivatives as P-glycoprotein inhibitors: molecular modeling, synthesis and sensitization of multidrug resistant cells to doxorubicin. European Journal of Medicinal Chemistry. 2020. Vol. 198. pp. 112331.
Grin M., Tikhonov S., Petrova A.S., Pogorilyy V., Noev A., Tatarskiy V.V., Shpakovsky D.B., Milaeva E.R., Kalinina E.V., Chernov N., Shtil A.A., Mironov A., Kaprin A., Filonenko E. New Derivatives of Bacteriopurpurin with Thiolated Au (I) Complexes: Dual Dark-and Light Activated Antitumor Potency. Anti-Cancer Agents in Medicinal Chemistry. 2020. Vol. 20. No. 1. pp. 49-58.
Anizon F., Giraud F., Ivanova E.S., Kaluzhny D.N., Shtil A., Cisnetti F., Moreau P. Synthesis and biological activities of new pyrrolocarbazole-imidazobenzimidazole conjugates. Tetrahedron Letters. 2020. Vol. 61. No. 30. pp. 152096.
Shtil A.A. Review of Patent Series eBook "Topics in Anti-Cancer Research, vol 6". Current Cancer Therapy Reviews. 2019. Vol. 15. No. 1. pp. 83.
High-Electron Density Nanomaterials for Theranostics
Roninson I.B., Gyorffy B., Mack Z.T., Shtil A.A., Shtutman M.S., Chen M., Broude E.V. Identifying cancers impacted by CDK8/19. Cells. 2019. Vol. 8. No. 8. pp. 821.
Petrova A.S., Olshevskaya V.A., Zaitsev A.V., Tatarsky V.V., Kalinina E.V., Andreev Y.A., Shtil A.A. New modified chlorin derivative as an antitumor photosensitizer: overcoming antioxidant defense in ovarian carcinoma cells sensitive and resistant to cisplatin. XIII International Conference "Synthesis and Application of Porphyrins and Their Analogues". 2019. pp. 54.
Belousov A.V., Morozov V.N., Krusanov G.A., Kolyvanova M.A., Shtil A.A. The Effect of Gold Nanoparticle Surface Modification with Polyethylene Glycol on the Absorbed Dose Distribution upon Irradiation with 137 Cs and 60 Co Photons. Biophysics. 2019. Vol. 64. No. 1. pp. 23–30.
Kalinina E.V., Andreev Y.A., Petrova A.S., Shtil A.A., Chernov N.N., Novichkova M.D., Nurmuradov N.K. Trx/TrxR system in redox-dependent regulation under development of cisplatin resistance in cancer cells. Free Radical Biology and Medicine. 2019. Vol. 139. No. 1. pp. 31.
Sosonyuk S.E., Peshich A., Tutushkina A.V., Khlevin D.A., Lozinskaya N.A., Gracheva Y.A., Glazunova V.A., Osolodkin D.I., Semenova M.N., Semenov V.V., Palyulin V.A., Proskurnina M.V., Shtil A.A., Zefirov N.S. Synthesis and cytotoxicity of novel simplified eleutherobin analogues as potential antitumour agents. Organic and Biomolecular Chemistry. 2019. Vol. 17. No. 10. pp. 2792-2797.
Yurkov D.I., Syromukov S.V., Tatarskiy V., Ivanova E.S., Khamidullina A.I., Yastrebova M.A., Sysoev V.I., Dobrov R.V., Belousov A.V., Morozov V.N., Kolyvanova M.A., Krusanov G.A., Zverev V.I., Shtil A.A. A Unique Prototypic Device for Radiation Therapy: The p53-Independent Antiproliferative Effect of Neutron Radiation. Acta Naturae (англоязычная версия). 2019. Vol. 11. No. 3(42). pp. 99-102.
Nuzhina J., Shtil A.A., Prilepskii A.Y., Vinogradov V.V. Preclinical Evaluation and Clinical Translation of Magnetite-Based Nanomedicines. Journal of Drug Delivery Science and Technology. 2019. Vol. 54. pp. 1773-2247.
Perevoshchikova K.A., Nichugovskiy A.I., Isagulieva A.K., Morozova N.G., Ivanov I.V., Maslov M.A., Shtil A.A. Synthesis of novel lipophilic tetraamines with cytotoxic activity. Mendeleev Communications. 2019. Vol. 29. No. 6. pp. 616-618.
Radchenko A.S., Kostyukov A.A., Markova A.A., Shtil A.A., Nekipelova T.D., Borissevitch I.E., Kuzmin V.A. Photoactivated biscarbocyanine dye with two conjugated chromophores: complexes with albumin, photochemical and phototoxic properties. Photochemical and Photobiological Sciences. 2019. Vol. 18. No. 10. pp. 2461-2468.
Новая комбинация неорганических композитов и органического соединения для элиминации клеток хронического миелоидного лейкоза
Ivanova E.S., Tatarskii V.V., Yastrebova M.A., Khamidullina A.I., Shunaev A.V., Kalinina A.A., Zeifman A.A., Novikov F.N., Dutikova Y.V., Chilov G.G., Shtil A.A. PF-114, a novel selective inhibitor of BCR-ABL tyrosine kinase, is a potent inducer of apoptosis in chronic myelogenous leukemia cells. International Journal of Oncology. 2019. Vol. 55. No. 1. pp. 289-297.
Dukhinova M.S., Prilepskii A.Y., Shtil A.A., Vinogradov V.V. Metal Oxide Nanoparticles in Therapeutic Regulation of Macrophage Functions. Nanomaterials. 2019. Vol. 9. No. 11. pp. 1631.
Rokitskaya T.I., Khailova L.S., Makarenkov A.V., Shunaev A.V., Tatarskiy V.V., Shtil A.A., Ol'Shevskaya V.A., Antonenko Y.N. Carborane derivatives of 1,2,3-triazole depolarize mitochondria by transferring protons through the lipid part of membranes. Biochimica et Biophysica Acta - Biomembranes. 2019. Vol. 1861. No. 3. pp. 573-583.
Ol'Shevskaya V.A., Alpatova V.M., Radchenko A.S., Tatarskii V.V., Ramonova A.A., Petrova A.S., Tatarskiy V.V., Zaitsev A.V., Kononova E.G., Ikonnikov N.S., Kostyukov A.A., Egorov A.E., Moisenovich M.M., Kuzmin V.A., Bragina N.A., Shtil A.A. Beta-Maleimide substituted meso-arylporphyrins: Synthesis, transformations, physico-chemical and antitumor properties. Dyes and Pigments. 2019. Vol. 171. pp. 107760.
Fakhardo A.F., Anastasova E.I., Gabdullina S.R., Solovyeva A.S., Saparova V.B., Chrishtop V.V., Koshevaya E.D., Krivoshapkina E.F., Krivoshapkin P.V., Kiselev G.O., Kalikina P.A., Koshel E.I., Shtil A.A., Vinogradov V.V. Toxicity Patterns of Clinically Relevant Metal Oxide Nanoparticles. ACS Applied Bio Materials. 2019. Vol. 2. No. 10. pp. 4427-4435.
Kuzmin V.A., Volnukhin V.A., Egorov A.E., Klimovich O.N., Kostyukov A.A., Nekipelova T.D., Khodot E.N., Shakhmatov V.V., Shevelev A.V., Shibaeva A.B., Shtil A.A. Furodihydroquinolines as Novel Photosensitizers for Photochemotherapy. Russian Journal of Physical Chemistry B. 2019. Vol. 13. No. 6. pp. 893-899.
Volodina Y.L., Dezhenkova L.G., Tikhomirov A.S., Tatarskii V.V., Kaluzhny D.N., Moisenovich A.M., Moisenovich M.M., Isagulieva A.K., Shtil A.A., Tsvetkov V., Shchekotikhin A.E. New anthra[2,3-b]furancarboxamides: a role of positioning of the carboxamide moiety in antitumor properties. European Journal of Medicinal Chemistry. 2019. Vol. 165. pp. 31-45.
The combination of copper oxide nanoparticles and N-acetylcysteine as a possible agent for chronic myeloid leukemia treatment
Kalinina E.V., Andreev Y.A., Lybova K., Hasan A.A., Petrova A.S., Chernov N.N., Shtil A.A., Novichkova M.D., Nurmuradov N.K. Thioredoxin/thioredoxin reductase system and redox-dependent regulation of adaptive antioxidant response under formation of cancer cell resistance to cisplatin. FEBS Open Bio. 2019. Vol. 9. No. S1. pp. 333.
High–Electron Density Nanomaterials for Theranostics
Belyaeva E.V., Markova A.A., Zakharko M.A., Radchenko A.S., Sigan A.L., Ikonnikov N.S., Shtil A.A., Chkanikov N.D. Chlorin Type Photosensitizers Soluble in Perfluorocarbons: Synthesis and Properties = Фотосенсибилизаторы хлоринового ряда, растворимые в перфторуглеродах: синтез и свойства. Fluorine Notes. 2019. No. 1(122). pp. 7-8.
Salakhova R.T., Pyatakov A.P., Zverev V.I., Pimentel B., Vivas R., Makarova L.A., Perov N.S., Tishin A.M., Shtil A.A., Reis M.S. The frequency dependence of magnetic heating for La0.75Sr0.25MnO3 nanoparticles. Journal of Magnetism and Magnetic Materials. 2019. Vol. 470. pp. 38-40.
Morozova N.G., Shmendel E.V., Timofeev G.A., Ivanov I.V., Kubasova T.S., Plyavnik N.V., Markova A.A., Maslov M.A., Shtil A.A. New design of cationic alkyl glycoglycerolipids toxic to tumor cells. Mendeleev Communications. 2019. Vol. 29. No. 2. pp. 166-168.
Antonenko T.A., Shtil A.A., Milaeva E.R. Coordination and Organometallic Compounds with 2,6-di-tert-butylphenol fragments. Synthesis, Structure and Biological Activity. Сборник тезисов всероссийского кластера конференций по неорганической химии "InorgChem2018". 2018. pp. 160.
Kalinina E.V., Andreev Y.A., Lubova K.I., Petrova A.S., Shtil A.A., Chernov N.N. Redox-dependent change in the expression of genes controlling cellular ROS/antioxidants balance under formation of cancer cell resistance to cisplatin. FEBS Open Bio. 2018. Vol. 8. No. S1. pp. 357.
Pimentel B., Caraballo-Vivas R.J., Checca N.R., Zverev V.I., Salakhova R.T., Makarova L.A., Pyatakov A.P., Perov N.S., Tishin A.M., Shtil A.A., Rossi A.L., Reis M.S. Threshold heating temperature for magnetic hyperthermia: controlling the heat exchange with the blocking temperature of magnetic nanoparticles. Journal of Solid State Chemistry. 2018. Vol. 260. pp. 34-38.
Morozov V.N., Belousov A.V., Krusanov G.A., Kolyvanova M.A., Chernyaev A.P., Shtil A.A. Secondary Electron Spectral Changes of Irradiated Gold Nanoparticle Caused By PEGylation. KnE Energy & Physics. 2018. pp. 278–282.
Shaikhutdinova N.D., Shaikhutdinov T.F., Frolov G.A., Borisova A.I., Akopdzhanov A.G., Shtil A.A. Design of nanodispersed magnetoactive systems for targeted drug delivery. Nanotechnologies in Russia. 2018. Vol. 13. No. 5-6. pp. 317-321.
Shtil A.A. Meet Our Sectional Editor. Anti-Cancer Agents in Medicinal Chemistry. 2018. Vol. 18. No. 12. pp. 1649.
Belousov A.V., Morozov V.N., Krusanov G.A., Kolyvanova M.A., Chernyaev A.P., Shtil A.A. Modeling the Effect of Surface Modification of Gold Nanoparticles Irradiated with Co-60 on the Secondary Particles Emission Spectrum. Doklady Physics. 2018. Vol. 63. No. 3. pp. 96-99.
Tikhomirov A.S., Lin C., Volodina Y.L., Dezhenkova L.G., Tatarskiy V.V., Schols D., Shtil A.A., Kaur P., Chueh P.J., Shchekotikhin A.E. New antitumor anthra[2,3-b]furan-3-carboxamides: Synthesis and structure-activity relationship. European Journal of Medicinal Chemistry. 2018. Vol. 148. pp. 128-139.
Vinogradov V.V., Drozdov A.S., Mingabudinova L.R., Shabanova E.M., Kolchina N.V., Anastasova E.I., Markova A.A., Shtil A.A., Milichko V.A., Starova G.L., Precker R., Vinogradov A.V., Hey-Hawkins E., Pidko E.A. Composites Based on Heparin and MIL-101(Fe): The Drug Releasing Depot for Anticoagulant Therapy and Advanced Medical Nanofabrication. Journal of Materials Chemistry B. 2018. Vol. 6. No. 16. pp. 2450-2459.
Belyaeva E.V., Markova A.A., Kaluzhny D.N., Sigan A.L., Gervitz L.L., Ataeva A.N., Chkanikov N.D., Shtil A.A. Novel Fluorinated Porphyrins Sensitize Tumor Cells to Photodamage in Normoxia and Hypoxia: Synthesis and Biocompatible Formulations. Anti-Cancer Agents in Medicinal Chemistry. 2018. Vol. 18. No. 4. pp. 617-627.
Douara B., Esvan Y.J., Pereira E., Giraud F., Volodina Y.L., Kaluzhny D.N., Shtil A.A., Anizon F., Moreau P. Synthesis and antiproliferative evaluation of glucosylated pyrazole analogs of K252c. Tetrahedron. 2018. Vol. 74. No. 8. pp. 892-901.
Tikhomirov A.S., Shtil A.A., Shchekotikhin A.E. Advances in the Discovery of Anthraquinone-Based Anticancer Agents. Recent Patents on Anti-cancer Drug Discovery. 2018. Vol. 13. No. 2. pp. 159-183.
Morozov V.N., Belousov A.V., Krusanov G.A., Kolyvanova M.A., Krivoshapkin P.V., Vinogradov V.V., Chernyaev A.P., Shtil A.A. Nanosized Particles of Tantalum, Hafnium, and Cerium Oxides Used with Monochromatic Photon Beams and Brachytherapy Sources. Optics and spectroscopy. 2018. Vol. 125. No. 1. pp. 104-106.
Морозов В.Н., Белоусов А.В., Крусанов Г.А., Колыванова М.А., Кривошапкин П.В., Виноградов В.В., Черняев А.П., Штиль А.А. Наноразмерные оксиды тантала, гафния и церия для монохроматических пучков фотонов и брахитерапии. Оптика и спектроскопия. 2018. Т. 125. № 1. С. 101-104.
Petrova A., Ol'Shevskaya V., Zaitsev A., Tatarskiy V.V., Kalinina E., Andreev Y., Chernov N., Shtil A.A. Antioxidant mechanisms in ovary adenocarcinoma cells resistant to cisplatin do not rescue from photonecrosis: implications for photodynamic therapy. FEBS Open Bio. 2018. Vol. 8. No. S1. pp. 214.
Lukasheva E.V., Kotovshchikov Y.N., Latyshev G.V., Kalinina E.V., Shtil A.A., Kolotova E.S., Lukashev N.V. Transition metals catalyzed reactions–a new approach to the aryl-, azolyl-and triazolylsubstituted steroids–active compounds against human MCF7 breast and SCOV3 ovarian carcinoma cells. FEBS Open Bio. 2018. Vol. 8. No. S1. pp. 238.
Saparova V.B., Shtil A.A. The role of 53-activators for combined cancer treatment. Альманах научных работ молодых ученых Университета ИТМО. 2018. Vol. 3. pp. 277-278.
Высокоэлектроноплотные наноматериалы для онкотераностики
Boron-Based Compounds: Potential and Emerging Applications in Medicine. Cp. 3.3. Carborane Derivatives of Porphyrins and Chlorins for Photodynamic and Boron Neutron Capture Therapies: Synthetic Strategies / Valentina A. Ol'shevskaya Andrei V. Zaitsev Alexander A. Shtil
Nadysум G., Tikhomirov A.S., Lin M., Yang Y., Dezhenkova L.G., Chen H., Kaluzhny D.N., Schols D., Shtil A.A., Shchekotikhin A.E., Chueh P.J. Aminomethylation of heliomycin: Preparation and anticancer characterization of the first series of semi-synthetic derivatives. European Journal of Medicinal Chemistry. 2018. Vol. 143. pp. 1553-1562.
Shpakovsky D.B., Shtil A.A., Kharitonashvili E.V., Tyurin V.Y., Antonenko T.A., Nazarov A.A., Osipova V.P., Berberova N.T., Foteeva L.S., Schmidt C., Ott I., Milaeva E.R. The antioxidant 2,6-di-tert-butylphenol moiety attenuates the pro-oxidant properties of the auranofin analogue. Metallomics. 2018. Vol. 10. No. 3. pp. 406-413.
Zverev V.I., Pyatakov A.P., Shtil A.A., Tishin A.M. Novel applications of magnetic materials and technologies for medicine. Journal of Magnetism and Magnetic Materials. 2018. Vol. 459. pp. 182-186.
Beniaminov A.D., Dezhenkova L.G., Mamaeva O.K., Shchyolkina A.K., Tevyashova A.N., Kaluzhny D.N., Shtil A.A. Divalent cations are dispensable for binding to DNA of a novel positively charged olivomycin A derivative. PLoS ONE. 2018. Vol. 13. No. 2. pp. e0191923.
Belousov A.V., Morozov V.N., Krusanov G.A., Kolyvanova M.A., Chernyaev A.P., Shtil A.A. Spectra of secondary particles generated upon virtual irradiation of gold nanosensitizers: Implications for surface modification. Biomedical Physics and Engineering Express. 2018. Vol. 4. No. 4. pp. 045023.
Prilepskii A.Y., Fakhardo A.F., Drozdov A.S., Vinogradov V.V., Dudanov I.P., Shtil A.A., Bel'Tyukov P., Shibeko A., Koltsova E., Nechipurenko D., Vinogradov V.V. Urokinase-conjugated magnetite nanoparticles as a promising drug delivery system for targeted thrombolysis: synthesis and preclinical evaluation. ACS Applied Materials and Interfaces. 2018. Vol. 10. No. 43. pp. 36764-36775.
Silva E.R., Pavanelli A.L., Mostaco L.B., Schaberle F.A., Galembeck S.E., Goncalves P.J., Costa E Silva R., Ferreira L.P., Nekipelova T.D., Kostyukov A.A., Radchenko A.S., Shtil A.A., Kuzmin V.A., Borissevitch I.E. Phototransformation of cyanine dye with two chromophores. Effects of oxygen and dye concentration. Journal of Photochemistry and Photobiology A: Chemistry. 2017. Vol. 349. pp. 42-48.
Shtil A.A., Miyoshi N., Karaya K., Shimada I., Tanaka H., Sakurai Y., Suzuki M., Zaitsev A.V., Ol’Shevskaya V., Rychkov G., Ono K., Kalinin V. Combination therapy of tumor model with pdt in radiological regions. Journal of International Scientific Publications: Materials, Methods and Technologies (Online). 2017. Vol. 11. pp. 395-402.
DNA nanomachines for targeting nucleic acids in cancer cells
PEGYLATION MODULATES THE SPECTRUM OF SECOND-ARY ELECTRONS UPON IRRADIATION OF GOLD NANO-PARTICLES: A MONTE-CARLO CALCULATION
Andreeva Y.I., Drozdov A.S., Fakhardo A.F., Cheplagin N.A., Shtil A.A., Vinogradov V.V. The controllable destabilization route for synthesis of low cytotoxic magnetic nanospheres with photonic response. Scientific Reports. 2017. Vol. 7. pp. 11343.
Kostyukov A.A., Pozdnyakova N.V., Shevelev A.B., Radchenko A.S., Golovina G.V., Klimovich O.N., Shtil’ A.A., Codognato D., Goncalves P., Pavanelli A., Ferreira L.P., Amado A.M., Borisevich Y.E., Kuzmin V.A. Complexes of alpha-fetoprotein and serum albumin with biscarbocyanine dye. High Energy Chemistry. 2017. Vol. 51. No. 3. pp. 233-235.
Shtil A.A., Ol'Shevskaya V.A., Zaitsev A.V., Radchenko A.S., Petrova A.S., Markova A.A., Miyoshi N., Borissevitch I.E., Kuzmin V.A. Chemical modifications of tetrapyrrole and carbocyanine scaffolds: On the road to optimized antitumor photosensitizers. Photodiagnosis and Photodynamic Therapy. 2017. Vol. 100. No. 17. pp. A24-A25.
Mechanisms of antioxidant protection and photoinduced death in cisplatin-sensitive and-resistant ovarian adenocarcinoma cells
Volkova Y.A., Chernoburova E.I., Petrova A.S., Shtil A.A., Zavarzin I.V. Reactions of hydrazones derived from oxamic acid thiohydrazides. Phosphorus, Sulfur and Silicon and the Related Elements. 2017. Vol. 192. No. 2. pp. 237-240.
Gornostaev L., Tsvetkov V., Markova A., Lavrikova T., Khalyavina Y., Kuznetsova A., Kaluzhny D., Shunayev A., Tsvetkova M., Glazunova V., Chernyshev V., Shtil A.A. The Oxime Derivatives of 1-R-1H-Naphtho[2,3-d][1,2,3]triazole-4,9-dione 2-oxides: Synthesis and Properties. Anti-Cancer Agents in Medicinal Chemistry. 2017. Vol. 17. No. 13. pp. 1814-1823.
Mechanisms of antioxidant protection and photoinduced death in cisplatin-sensitive and-resistant ovarian adenocarcinoma cells
Kostyukov A.A., Nekipelova T.D., Radchenko A.S., Golovina G.V., Klimovich O.N., Shtil A.A., Codognato D., Goncalves P., Pavanelli A., Ferreira L.P., Amado A.M., Borisevich Y.E., Kuzmin V.A. Triplet states of the complexes of biscarbocyanine dye with albumin. High Energy Chemistry. 2017. Vol. 51. No. 2. pp. 148-150.
Vasilyeva S.V., Shtil A.A., Petrova A.S., Balakhnin S.M., Achigecheva P.Y., Stetsenko D.A., Silnikov V.N. Conjugates of phosphorylated zalcitabine and lamivudine with SiO2 nanoparticles: Synthesis by CuAAC click chemistry and preliminary assessment of anti-HIV and antiproliferative activity. Bioorganic and Medicinal Chemistry. 2017. Vol. 25. No. 5. pp. 1696-1702.
Tishin A.M., Shtil A.A., Pyatakov A.P., Zverev V.I. Developing antitumor magnetic hyperthermia: Principles, materials and devices. Recent Patents on Anti-cancer Drug Discovery. 2016. Vol. 11. No. 4. pp. 360-375.
Российская Федерация, Санкт-Петербург
Российская Федерация, Санкт-Петербург