Штиль Александр Альбертович

Штиль Александр Альбертович
доктор медицинских наук
доцент (квалификационная категория "доцент практики"), химико-биологический кластер

Педагогический стаж

Общий стаж:
21 год

Публикации

122
Статья
2024 год

Цымбал С.А. The Copper Reduction Potential Determines the Reductive Cytotoxicity: Relevance to the Design of Metal–Organic Antitumor Drugs. MDPI. 2024. Vol. 29. No. 5. pp. 1032.

Статья
2023 год

Rusina P., Lisov A., Denisova A., Gandalipov E.R., Novikov F., Shtil A.A. Clinical CDK2 Inhibitors: Trends to Selectivity and Efficacy. Recent Patents on Anti-cancer Drug Discovery. 2023. Vol. 18. No. 2. pp. 102-107.

Статья
2023 год

Guk D., Gibadullina K.R., Burlutskiy R.O., Pavlov K.G., Moiseeva A., Tafeenko V.A., Lyssenko K.A., Gandalipov E.R., Shtil A., Beloglazkina E. New Titanocene (IV) Dicarboxylates with Potential Cytotoxicity: Synthesis, Structure, Stability and Electrochemistry. International Journal of Molecular Sciences. 2023. Vol. 24. No. 4. pp. 3340.

Статья
2023 год

Kokinos E.K., Tsymbal S.A., Galochkina A.V., Bezlepkina S.A., Nikolaeva J.V., Vershinina S.O., Shtro A., Tatarskiy V.V., Shtil A.A., Broude E.V., Roninson I.B., Dukhinova M. Inhibition of Cyclin-Dependent Kinases 8/19 Restricts Bacterial and Virus-Induced Inflammatory Responses in Monocytes. Viruses. 2023. Vol. 15. No. 6. pp. 1292.

Статья
2023 год

Kuchur O.A., Zavisrskiy A.V., Shtil А. Transcriptional Reprogramming Regulates Tumor Cell Survival in Response to Ionizing Radiation: a Role of p53. Bulletin of Experimental Biology and Medicine. 2023. Vol. 174. No. 5. pp. 659-665.

Тезисы
2023 год

Моделирование резистентности хронического миелоидного лейкоза к ингибиторам BCR-ABL в костном мозге

Статья
2022 год

Кокинос Е.К., Кузьмина Д., Кучур О.А., Цымбал С.А., Василичин В.А., Галочкина А.В., Завирский А.В., Башарин В.А., Штро А.А., Штиль А.А., Духинова М.С. Фенотипический и функциональный анализ линии моноцитов THP-1 как модели воспаления [Phenotypic and functional characteristic analysis of THP-1 cell line as a model of inflammation]. Иммунология [Immunologiya]. 2022. Т. 43. № 3. С. 277-287.

Тезисы
2022 год

Механизмы гибели опухолевых клеток при действии производных териндолона

Тезисы
2022 год

СИНТЕТИЧЕСКАЯ ЛЕТАЛЬНОСТЬ КЛЕТОК MYCN ПОЛОЖИТЕЛЬНОЙ НЕЙРОБЛАСТОМЫ ПОД ДЕЙСТВИЕМ СЕЛЕКТИВНЫХ ИНГИБИТОРОВ CDK2

Тезисы
2022 год

Определение цитотоксической и противоопухолевой активности комбинации медьорганических соединений и N-ацетилцистеина на модели полостных метастазов in vivo

Тезисы
2022 год

Ингибирование СDK8/19-зависимого перепрограммирования транскрипции - новый механизм радиосенситизации p53-положительных опухолевых клеток

Статья
2022 год

Цымбал С.А., Штиль А.А. Исследование переносимости медьсодержащих соединений и восстановителя для разработки модели терапии опухолевого асцита. Вопросы онкологии [Voprosy Onkologii]. 2022. Т. 68. № S3. С. 361-362.

Статья
2022 год

Ivanov V., Agamennone M., Iusupov I.R., Laghezza A., Novoselov A.M., Manasova E.V., Altieri A., Tortorella P., Shtil А., Kurkin A.V. Het(aryl)isatin to het(aryl)aminoindoline scaffold hopping: A route to selective inhibitors of matrix metalloproteinases. Arabian Journal of Chemistry. 2022. Vol. 15. No. 1. pp. 103492.

Статья
2021 год

Kuchur O.A., Kuzmina D., Dukhinova M.S., Shtil A. The p53 Protein Family in the Response of Tumor Cells to Ionizing Radiation: Problem Development. Acta Naturae (англоязычная версия). 2021. Vol. 13. No. 3. pp. 65-76.

Тезисы
2021 год

РОЛЬ СТАТУСА Р53 В ОТВЕТЕ ОПУХОЛЕВЫХ КЛЕТОК НА ИОНИЗИРУЮЩЕЕ ИЗЛУЧЕНИЕ ПРИ ИНГИБИРОВАНИИ CDK8/19

Статья
2021 год

Kuchur O.A., Kuchur P.D., Kuzmina D., Zavirsky A.V., Shtil A. Differential Regulation of BBC3/PUMA and PMAIP1/Noxa in Ionizing Radiation: the Role of p53. Cell and Tissue Biology. 2021. Vol. 15. No. 6. pp. 544-553.

Статья
2021 год

Bruter А., Rodionova M., Varlamova Е., Shtil А. Super-Enhancers in the Regulation of Gene Transcription: General Aspects and Antitumor Targets. Acta Naturae (англоязычная версия). 2021. Vol. 13. No. 1. pp. 4-15.

Тезисы
2021 год

Механизмы усиления гибели опухолевых клеток при ионизирующем излучении: связь между p53 и CDK8/19

Статья
2021 год

Кучур О.А., Кучур П.Д., Кузьмина Д.О., Завирский А.В., Штиль А.А. Дифференциальная регуляция BBC3/PUMA и PMAIP1/Noxa при ионизирующем излучении: роль p53 [Differential Regulation of BBC3/PUMA and PMAIP1/Noxa by Ionizing Radiation: A Role for p53]. Цитология [Tsitologiya]. 2021. Т. 63. № 4. С. 363-372.

Статья
2021 год

Tsymbal S., Agadzhanyan N., Shtil А. Oxidative stress associated with Cu2+to Cu+ reduction for eradicating wild type and multidrug-resistant tumor cells. Annals of Oncology. 2021. Vol. 32. No. Suppl.6. pp. S1365-S1365.

Статья
2021 год

Kuchur O.A., Zavirskiy A.V., Shtil А. Attenuation of p53 signaling by CDK8/19 sensitizes tumor cells to ionizing radiation. Annals of Oncology. 2021. Vol. 32. No. Suppl.6. pp. S1358-S1358.

Статья
2021 год

Medvedeva G., Kuzmina D., Nuzhina J.V., Shtil A.A., Dukhinova M.S. How macrophages become transcriptionally dysregulated: A hidden impact of antitumor therapy. International Journal of Molecular Sciences. 2021. Vol. 22. No. 5. pp. 2662.

Статья
2021 год

Брутер А.В., Родионова М.Д., Варламова Е.А., Штиль А.А. Суперэнхансеры в регуляции транскрипции генов: общебиологические аспекты и мишени противоопухолевой терапии. Acta Naturae (русскоязычная версия). 2021. Т. 13. № 1. С. 4-15.

Статья
2021 год

Кучур О.А., Кузьмина Д.О., Духинова М.С., Штиль А.А. Белки семейства p53 в ответе опухолевых клеток на ионизирующее излучение: развитие проблемы. Acta Naturae (русскоязычная версия). 2021. Т. 13. № 3. С. 65-76.

Тезисы
2021 год

Использование меди N-ацетилцистеином и аскорбатом для преодоления лекарственной устойчивости опухолевых клеток

Тезисы
2021 год

Attenuation of p53 signaling by CDK8/19 sensitizes tumor cells to ionizing radiation

Тезисы
2021 год

ИНГИБИРОВАНИЕ p53 ЧЕРЕЗ CDK8/19 ПОВЫШАЕТ ЧУВСТВИТЕЛЬНОСТЬ ОПУХОЛЕВЫХ КЛЕТОК К ИОНИЗИРУЮЩЕМУ ИЗЛУЧЕНИЮ

Тезисы
2021 год

65P - Oxidative stress associated with Cu2+ to Cu+ reduction for eradicating wild type and multidrug resistant tumor cells

Статья
2021 год

Tsymbal S.A., Moiseeva A., Agadzhanian N., Efimova S., Markova A.A., Guk D., Krasnovskaya O., Alpatova V., Zaitsev A.V., Shibaeva A., Tatarskiy V.V., Dukhinova M.S., Ol’Shevskaya V., Ostroumova O., Beloglazkina E., Shtil А. Copper-Containing Nanoparticles and Organic Complexes: Metal Reduction Triggers Rapid Cell Death via Oxidative Burst. International Journal of Molecular Sciences. 2021. Vol. 22. No. 20. pp. 11065.

Статья
2021 год

Shutkov I., Okulova Y.N., Tyurin V.Y., Sokolova E.V., Babkov D.A., Spasov A.A., Gracheva Y.A., Schmidt G., Kirsanov K., Shtil А., Redkozubova O., Shevtsova E.F., Milaeva E.R., Ott I., Nazarov A.A. Ru (III) Complexes with lonidamine-modified ligands. International Journal of Molecular Sciences. 2021. Vol. 22. No. 24. pp. 13468.

Статья
2020 год

Belousov A.V., Morozov V.N., Krusanov G.A., Moiseev A.N., Davydov A.S., Shtil A.A., Klimanov V.A., Kolyvanova M.A., Samoylov A.S. The Change in the Linear Energy Transfer of a Clinical Proton Beam in the Presence of Gold Nanoparticles. Biophysics. 2020. Vol. 65. No. 4. pp. 541-547.

Статья
2020 год

Vasilyeva S.V., Petrova A.S., Shtil A.A., Stetsenko D.A. Application of silicon dioxide nanoparticles modified with tumor-targeting ligands for cellular delivery of nucleoside triphosphate analogues. Journal of Saudi Chemical Society. 2020. Vol. 24. No. 1. pp. 98-104.

Тезисы
2020 год

Молекулярные механизмы чувствительности опухолевых клеток к терапевтическому ионизирующему излучению: p53 и CDK8/19

Тезисы
2020 год

Комбинированное применение наночастиц оксида меди и N-ацетилцистеина для преодоления лекарственной устойчивости опухолевых клеток

Тезисы
2020 год

PHOTOCURABLE FILMS BASED ON FIBROIN AND GELATIN FOR REGENERATION OF SKIN COVER

Статья
2020 год

Grin M., Tikhonov S., Petrova A.S., Pogorilyy V., Noev A., Tatarskiy V.V., Shpakovsky D.B., Milaeva E.R., Kalinina E.V., Chernov N., Shtil A.A., Mironov A., Kaprin A., Filonenko E. New Derivatives of Bacteriopurpurin with Thiolated Au (I) Complexes: Dual Dark-and Light Activated Antitumor Potency. Anti-Cancer Agents in Medicinal Chemistry. 2020. Vol. 20. No. 1. pp. 49-58.

Тезисы
2020 год

The role of p53 status in response to ionizing radiation

Монография
2020 год

Boron-Based Compounds: Potential and Emerging Applications in Medicine

Статья
2020 год

Bessonov I., Moysenovich A., Arkhipova A., Ezernitskaya M., Efremov Y., Solodilov V., Timashev P., Shaytan K., Shtil A., Moisenovich M. The mechanical properties, secondary structure, and osteogenic activity of photopolymerized fibroin. Polymers. 2020. Vol. 12. No. 3. pp. 646.

Статья
2020 год

Tikhomirov A.S., Litvinova V., Andreeva D.V., Tsvetkov V., Dezhenkova L.G., Volodina Y.L., Kaluzhny D.N., Treshalin I., Schols D., Ramonova A.A., Moisenovich M.M., Shtil A.A., Shchekotikhin A.E. Amides of pyrrole- and thiophene-fused anthraquinone derivatives: A role of the heterocyclic core in antitumor properties. European Journal of Medicinal Chemistry. 2020. Vol. 199. pp. 112294.

Статья
2020 год

Moysenovich A.M., Tatarskiy V.V., Yastrebova M.A., Bessonov I.V., Arkhipova A.Y., Kolosov A.S., Davydova L.I., Khamidullina A.I., Bogush V.G., Debabov V.G., Shaitan K.V., Shtil A.A., Moisenovich M.M. Akt and Src mediate the photocrosslinked fibroin-induced neural differentiation. NeuroReport. 2020. Vol. 31. No. 10. pp. 770–775.

Статья
2020 год

Anizon F., Giraud F., Ivanova E.S., Kaluzhny D.N., Shtil A., Cisnetti F., Moreau P. Synthesis and biological activities of new pyrrolocarbazole-imidazobenzimidazole conjugates. Tetrahedron Letters. 2020. Vol. 61. No. 30. pp. 152096.

Статья
2020 год

Morozov K.V., Kolyvanova M.A., Kartseva M.E., Shishmakova E.M., Dement’Eva O.V., Isagulieva A.K., Salpagarov M.H., Belousov A.V., Rudoy V.M., Shtil A.A., Samoylov A.S., Morozov V.N. Radiosensitization by gold nanoparticles: impact of the size, dose rate, and photon energy. Nanomaterials. 2020. Vol. 10. No. 5. pp. 952.

Статья
2020 год

Markova A.A., Belyaeva E.V., Radchenko A.S., Dmitrieva M.V., Sigan A.L., Shtil A.A., Chkanikov N.D. Perfluorocarbon nanoemulsions containing fluorinated photosensitizer for photodynamic cancer therapy. IOP Conference Series: Materials Science and Engineering. 2020. Vol. 848. No. 1. pp. 012054.

Статья
2020 год

Kostyukov A.A., Egorov A.E., Mestergazi M.G., Shmykova A.M., Podrugina T.A., Borissevitch I.E., Shtil A.A., Kuzmin V.A. Photochemical properties of new bis-cyanine dye as a promising agent for in vivo imaging. Mendeleev Communications. 2020. Vol. 30. No. 4. pp. 442-444.

Статья
2020 год

Silaeva Y.Y., Kalmykov V.A., Varlamova E.A., Korshunov E.N., Korshunova D.S., Kubekina M.V., Shtil A.A., Roninson I.B., Deykin A.V. Genome editing as an approach to the study of in vivo transcription reprogramming. Doklady Biochemistry and Biophysics. 2020. Vol. 490. No. 1. pp. 43-46.

Статья
2020 год

Gornostaev L.M., Fominykh O.I., Rukovets T.A., Lavrikova T.I., Khalyavina J.G., Shtil A.A., Shunaev A.V., Dunaev S.F., Murashova E.V., Chernyshev V.V. Synthesis of 6b, 11b-dihydroxy-12-methylphenyl-11b, 12-dihydrobenzo-[g] indeno [1, 2-b] indole-5, 6, 7 (6b H)-triones and 2-(3-hydroxy-4, 9-dioxo-4, 9-dihydro-1 H-benzo [f] indol-2-yl) benzamides, their structure and antiproliferative activity. Chemistry of Heterocyclic Compounds. 2020. Vol. 56. No. 1. pp. 47-54.

Статья
2020 год

Kotliarova M.S., Soldatenko A.S., Arkhipova A.Y., Bessonov I.V., Davydova L.I., Moysenovich A.M., Bogush V.G., Debabov V.G., Shtil A.A., Moisenovich M.M., Shaitan K.V. Photocurable Films Based on Fibroin and Gelatin for Skin Regeneration. Moscow University Biological Sciences Bulletin. 2020. Vol. 75. No. 1. pp. 20-25.

Статья
2020 год

Beniaminov A.D., Chashchina G.V., Livshits M.A., Kechko O.I., Mitkevich V.A., Mamaeva O.K., Tevyashova A.N., Shtil A.A., Shchyolkina A.K., Kaluzhny D.N. Discrimination between G/C Binding Sites by Olivomycin A Is Determined by Kinetics of the Drug-DNA Interaction. International Journal of Molecular Sciences. 2020. Vol. 21. No. 15. pp. 5299.

Статья
2020 год

Gornostaev L.M., Fominykh O.I., Rukovets T.A., Lavrikova T.I., Khalyavina J.G., Shtil A., Shunaev A.V., Dunaev S.F., Murashova E.V., Chernyshev V.V. Synthesis of 6b,11b-dihydroxy-12-methylphenyl-11b,12-dihydrobenzo- [g]indeno[1,2-b]indole-5,6,7(6bH)-triones and 2-(3-hydroxy-4,9-dioxo-4,9-dihydro-1H-benzo[f]indol-2-yl)benzamides, their structure and antiproliferative activity. Chemistry of Heterocyclic Compounds. 2020. Vol. 56. No. 1. pp. 47-54.

Статья
2020 год

Marsova M., Odorskaya M., Novichkova M., Polyakova V., Abilev S., Kalinina E., Shtil A., Poluektova E., Danilenko V. The Lactobacillus brevis 47 f strain protects the murine intestine from enteropathy induced by 5-fluorouracil. Microorganisms. 2020. Vol. 8. No. 6. pp. 876.

Статья
2020 год

Sagnou M., Novikov F.N., Ivanova E.S., Alexiou P., Stroylov V.S., Titov I.Y., Tatarskiy V., Vagida M.S., Pelecanou M., Shtil A.A., Chilov G.G. Novel curcumin derivatives as P-glycoprotein inhibitors: molecular modeling, synthesis and sensitization of multidrug resistant cells to doxorubicin. European Journal of Medicinal Chemistry. 2020. Vol. 198. pp. 112331.

Статья
2020 год

Dukhinova M.S., Shestovskaya M.V., Shtil A.A. Metal Nanoparticles in Immunotherapy: Applications, Limitations and Pespectives. Research & Development in Material Science. 2020. Vol. 12(4). No. 3. pp. 1292-1295.

Статья
2020 год

Morozov V.N., Belousov A.V., Zverev V.I., Shtil A.A., Kolyvanova M.A., Krivoshapkin P.V. The Prospects of Metal Oxide Nanoradiosensitizers: The Effect of the Elemental Composition of Particles and Characteristics of Radiation Sources on Enhancement of the Adsorbed Dose. Biophysics. 2020. Vol. 65. No. 4. pp. 533-540.

Статья
2020 год

Kuchur O.A., Tsymbal S.A., Shestovskaya M.V., Serov N.S., Dukhinova M.S., Shtil A.A. Metal-derived nanoparticles in tumor theranostics: Potential and limitations. Journal of Inorganic Biochemistry. 2020. Vol. 209. pp. 111117.

Статья
2020 год

Vasilichin V.A., Tsymbal S.A., Fakhardo A.F., Anastasova E., Marchenko A.S., Shtil A., Vinogradov V.V., Koshel E. Effects of Metal Oxide Nanoparticles on Toll-Like Receptor mRNAs in Human Monocytes. Nanomaterials. 2020. Vol. 10. No. 1. pp. 127.

Статья
2020 год

Moysenovich A.M., Moisenovich M.M., Sudina A.K., Tatarskiy V., Khamidullina A.I., Yastrebova M.A., Davydova L.I., Bogush V.G., Debabov V.G., Arkhipova A.Y., Shaitan K.V., Shtil A.A., Demina I.A. Recombinant Spidroin Films Attenuate Individual Markers of Glucose Induced Aging in NIH 3T3 Fibroblasts. Biochemistry (Moscow). 2020. Vol. 85. No. 7. pp. 808–819.

Тезисы
2020 год

Single vs Multiple Drug Targets: Revising the Therapeutic Concept to Combat Intractable Cancers

Статья
2019 год

Yurkov D.I., Syromukov S.V., Tatarskiy V., Ivanova E.S., Khamidullina A.I., Yastrebova M.A., Sysoev V.I., Dobrov R.V., Belousov A.V., Morozov V.N., Kolyvanova M.A., Krusanov G.A., Zverev V.I., Shtil A.A. A Unique Prototypic Device for Radiation Therapy: The p53-Independent Antiproliferative Effect of Neutron Radiation. Acta Naturae (англоязычная версия). 2019. Vol. 11. No. 3(42). pp. 99-102.

Тезисы
2019 год

The combination of copper oxide nanoparticles and N-acetylcysteine as a possible agent for chronic myeloid leukemia treatment

Статья
2019 год

Ivanova E.S., Tatarskii V.V., Yastrebova M.A., Khamidullina A.I., Shunaev A.V., Kalinina A.A., Zeifman A.A., Novikov F.N., Dutikova Y.V., Chilov G.G., Shtil A.A. PF-114, a novel selective inhibitor of BCR-ABL tyrosine kinase, is a potent inducer of apoptosis in chronic myelogenous leukemia cells. International Journal of Oncology. 2019. Vol. 55. No. 1. pp. 289-297.

Тезисы
2019 год

Новая комбинация неорганических композитов и органического соединения для элиминации клеток хронического миелоидного лейкоза

Тезисы
2019 год

High-Electron Density Nanomaterials for Theranostics

Тезисы
2019 год

High–Electron Density Nanomaterials for Theranostics

Статья
2019 год

Perevoshchikova K.A., Nichugovskiy A.I., Isagulieva A.K., Morozova N.G., Ivanov I.V., Maslov M.A., Shtil A.A. Synthesis of novel lipophilic tetraamines with cytotoxic activity. Mendeleev Communications. 2019. Vol. 29. No. 6. pp. 616-618.

Статья
2019 год

Petrova A.S., Olshevskaya V.A., Zaitsev A.V., Tatarsky V.V., Kalinina E.V., Andreev Y.A., Shtil A.A. New modified chlorin derivative as an antitumor photosensitizer: overcoming antioxidant defense in ovarian carcinoma cells sensitive and resistant to cisplatin. XIII International Conference "Synthesis and Application of Porphyrins and Their Analogues". 2019. pp. 54.

Статья
2019 год

Belousov A.V., Morozov V.N., Krusanov G.A., Kolyvanova M.A., Shtil A.A. The Effect of Gold Nanoparticle Surface Modification with Polyethylene Glycol on the Absorbed Dose Distribution upon Irradiation with 137 Cs and 60 Co Photons. Biophysics. 2019. Vol. 64. No. 1. pp. 23–30.

Статья
2019 год

Roninson I.B., Gyorffy B., Mack Z.T., Shtil A.A., Shtutman M.S., Chen M., Broude E.V. Identifying cancers impacted by CDK8/19. Cells. 2019. Vol. 8. No. 8. pp. 821.

Статья
2019 год

Shtil A.A. Review of Patent Series eBook "Topics in Anti-Cancer Research, vol 6". Current Cancer Therapy Reviews. 2019. Vol. 15. No. 1. pp. 83.

Статья
2019 год

Morozova N.G., Shmendel E.V., Timofeev G.A., Ivanov I.V., Kubasova T.S., Plyavnik N.V., Markova A.A., Maslov M.A., Shtil A.A. New design of cationic alkyl glycoglycerolipids toxic to tumor cells. Mendeleev Communications. 2019. Vol. 29. No. 2. pp. 166-168.

Статья
2019 год

Kalinina E.V., Andreev Y.A., Petrova A.S., Shtil A.A., Chernov N.N., Novichkova M.D., Nurmuradov N.K. Trx/TrxR system in redox-dependent regulation under development of cisplatin resistance in cancer cells. Free Radical Biology and Medicine. 2019. Vol. 139. No. 1. pp. 31.

Статья
2019 год

Salakhova R.T., Pyatakov A.P., Zverev V.I., Pimentel B., Vivas R., Makarova L.A., Perov N.S., Tishin A.M., Shtil A.A., Reis M.S. The frequency dependence of magnetic heating for La0.75Sr0.25MnO3 nanoparticles. Journal of Magnetism and Magnetic Materials. 2019. Vol. 470. pp. 38-40.

Статья
2019 год

Ol'Shevskaya V.A., Alpatova V.M., Radchenko A.S., Tatarskii V.V., Ramonova A.A., Petrova A.S., Tatarskiy V.V., Zaitsev A.V., Kononova E.G., Ikonnikov N.S., Kostyukov A.A., Egorov A.E., Moisenovich M.M., Kuzmin V.A., Bragina N.A., Shtil A.A. Beta-Maleimide substituted meso-arylporphyrins: Synthesis, transformations, physico-chemical and antitumor properties. Dyes and Pigments. 2019. Vol. 171. pp. 107760.

Статья
2019 год

Radchenko A.S., Kostyukov A.A., Markova A.A., Shtil A.A., Nekipelova T.D., Borissevitch I.E., Kuzmin V.A. Photoactivated biscarbocyanine dye with two conjugated chromophores: complexes with albumin, photochemical and phototoxic properties. Photochemical and Photobiological Sciences. 2019. Vol. 18. No. 10. pp. 2461-2468.

Статья
2019 год

Kalinina E.V., Andreev Y.A., Lybova K., Hasan A.A., Petrova A.S., Chernov N.N., Shtil A.A., Novichkova M.D., Nurmuradov N.K. Thioredoxin/thioredoxin reductase system and redox-dependent regulation of adaptive antioxidant response under formation of cancer cell resistance to cisplatin. FEBS Open Bio. 2019. Vol. 9. No. S1. pp. 333.

Статья
2019 год

Belyaeva E.V., Markova A.A., Zakharko M.A., Radchenko A.S., Sigan A.L., Ikonnikov N.S., Shtil A.A., Chkanikov N.D. Chlorin Type Photosensitizers Soluble in Perfluorocarbons: Synthesis and Properties = Фотосенсибилизаторы хлоринового ряда, растворимые в перфторуглеродах: синтез и свойства. Fluorine Notes. 2019. No. 1(122). pp. 7-8.

Статья
2019 год

Kuzmin V.A., Volnukhin V.A., Egorov A.E., Klimovich O.N., Kostyukov A.A., Nekipelova T.D., Khodot E.N., Shakhmatov V.V., Shevelev A.V., Shibaeva A.B., Shtil A.A. Furodihydroquinolines as Novel Photosensitizers for Photochemotherapy. Russian Journal of Physical Chemistry B. 2019. Vol. 13. No. 6. pp. 893-899.

Статья
2019 год

Fakhardo A.F., Anastasova E.I., Gabdullina S.R., Solovyeva A.S., Saparova V.B., Chrishtop V.V., Koshevaya E.D., Krivoshapkina E.F., Krivoshapkin P.V., Kiselev G.O., Kalikina P.A., Koshel E.I., Shtil A.A., Vinogradov V.V. Toxicity Patterns of Clinically Relevant Metal Oxide Nanoparticles. ACS Applied Bio Materials. 2019. Vol. 2. No. 10. pp. 4427-4435.

Статья
2019 год

Nuzhina J., Shtil A.A., Prilepskii A.Y., Vinogradov V.V. Preclinical Evaluation and Clinical Translation of Magnetite-Based Nanomedicines. Journal of Drug Delivery Science and Technology. 2019. Vol. 54. pp. 1773-2247.

Статья
2019 год

Dukhinova M.S., Prilepskii A.Y., Shtil A.A., Vinogradov V.V. Metal Oxide Nanoparticles in Therapeutic Regulation of Macrophage Functions. Nanomaterials. 2019. Vol. 9. No. 11. pp. 1631.

Статья
2019 год

Rokitskaya T.I., Khailova L.S., Makarenkov A.V., Shunaev A.V., Tatarskiy V.V., Shtil A.A., Ol'Shevskaya V.A., Antonenko Y.N. Carborane derivatives of 1,2,3-triazole depolarize mitochondria by transferring protons through the lipid part of membranes. Biochimica et Biophysica Acta - Biomembranes. 2019. Vol. 1861. No. 3. pp. 573-583.

Статья
2019 год

Volodina Y.L., Dezhenkova L.G., Tikhomirov A.S., Tatarskii V.V., Kaluzhny D.N., Moisenovich A.M., Moisenovich M.M., Isagulieva A.K., Shtil A.A., Tsvetkov V., Shchekotikhin A.E. New anthra[2,3-b]furancarboxamides: a role of positioning of the carboxamide moiety in antitumor properties. European Journal of Medicinal Chemistry. 2019. Vol. 165. pp. 31-45.

Статья
2019 год

Sosonyuk S.E., Peshich A., Tutushkina A.V., Khlevin D.A., Lozinskaya N.A., Gracheva Y.A., Glazunova V.A., Osolodkin D.I., Semenova M.N., Semenov V.V., Palyulin V.A., Proskurnina M.V., Shtil A.A., Zefirov N.S. Synthesis and cytotoxicity of novel simplified eleutherobin analogues as potential antitumour agents. Organic and Biomolecular Chemistry. 2019. Vol. 17. No. 10. pp. 2792-2797.

Статья
2018 год

Shpakovsky D.B., Shtil A.A., Kharitonashvili E.V., Tyurin V.Y., Antonenko T.A., Nazarov A.A., Osipova V.P., Berberova N.T., Foteeva L.S., Schmidt C., Ott I., Milaeva E.R. The antioxidant 2,6-di-tert-butylphenol moiety attenuates the pro-oxidant properties of the auranofin analogue. Metallomics. 2018. Vol. 10. No. 3. pp. 406-413.

Статья
2018 год

Saparova V.B., Shtil A.A. The role of 53-activators for combined cancer treatment. Альманах научных работ молодых ученых Университета ИТМО. 2018. Vol. 3. pp. 277-278.

Статья
2018 год

Beniaminov A.D., Dezhenkova L.G., Mamaeva O.K., Shchyolkina A.K., Tevyashova A.N., Kaluzhny D.N., Shtil A.A. Divalent cations are dispensable for binding to DNA of a novel positively charged olivomycin A derivative. PLoS ONE. 2018. Vol. 13. No. 2. pp. e0191923.

Статья
2018 год

Tikhomirov A.S., Lin C., Volodina Y.L., Dezhenkova L.G., Tatarskiy V.V., Schols D., Shtil A.A., Kaur P., Chueh P.J., Shchekotikhin A.E. New antitumor anthra[2,3-b]furan-3-carboxamides: Synthesis and structure-activity relationship. European Journal of Medicinal Chemistry. 2018. Vol. 148. pp. 128-139.

Статья
2018 год

Shtil A.A. Meet Our Sectional Editor. Anti-Cancer Agents in Medicinal Chemistry. 2018. Vol. 18. No. 12. pp. 1649.

Статья
2018 год

Tikhomirov A.S., Shtil A.A., Shchekotikhin A.E. Advances in the Discovery of Anthraquinone-Based Anticancer Agents. Recent Patents on Anti-cancer Drug Discovery. 2018. Vol. 13. No. 2. pp. 159-183.

Монография
2018 год

Boron-Based Compounds: Potential and Emerging Applications in Medicine. Cp. 3.3. Carborane Derivatives of Porphyrins and Chlorins for Photodynamic and Boron Neutron Capture Therapies: Synthetic Strategies / Valentina A. Ol'shevskaya Andrei V. Zaitsev Alexander A. Shtil

Статья
2018 год

Douara B., Esvan Y.J., Pereira E., Giraud F., Volodina Y.L., Kaluzhny D.N., Shtil A.A., Anizon F., Moreau P. Synthesis and antiproliferative evaluation of glucosylated pyrazole analogs of K252c. Tetrahedron. 2018. Vol. 74. No. 8. pp. 892-901.

Статья
2018 год

Морозов В.Н., Белоусов А.В., Крусанов Г.А., Колыванова М.А., Кривошапкин П.В., Виноградов В.В., Черняев А.П., Штиль А.А. Наноразмерные оксиды тантала, гафния и церия для монохроматических пучков фотонов и брахитерапии. Оптика и спектроскопия. 2018. Т. 125. № 1. С. 101-104.

Статья
2018 год

Morozov V.N., Belousov A.V., Krusanov G.A., Kolyvanova M.A., Krivoshapkin P.V., Vinogradov V.V., Chernyaev A.P., Shtil A.A. Nanosized Particles of Tantalum, Hafnium, and Cerium Oxides Used with Monochromatic Photon Beams and Brachytherapy Sources. Optics and spectroscopy. 2018. Vol. 125. No. 1. pp. 104-106.

Статья
2018 год

Belyaeva E.V., Markova A.A., Kaluzhny D.N., Sigan A.L., Gervitz L.L., Ataeva A.N., Chkanikov N.D., Shtil A.A. Novel Fluorinated Porphyrins Sensitize Tumor Cells to Photodamage in Normoxia and Hypoxia: Synthesis and Biocompatible Formulations. Anti-Cancer Agents in Medicinal Chemistry. 2018. Vol. 18. No. 4. pp. 617-627.

Статья
2018 год

Vinogradov V.V., Drozdov A.S., Mingabudinova L.R., Shabanova E.M., Kolchina N.V., Anastasova E.I., Markova A.A., Shtil A.A., Milichko V.A., Starova G.L., Precker R., Vinogradov A.V., Hey-Hawkins E., Pidko E.A. Composites Based on Heparin and MIL-101(Fe): The Drug Releasing Depot for Anticoagulant Therapy and Advanced Medical Nanofabrication. Journal of Materials Chemistry B. 2018. Vol. 6. No. 16. pp. 2450-2459.

Статья
2018 год

Belousov A.V., Morozov V.N., Krusanov G.A., Kolyvanova M.A., Chernyaev A.P., Shtil A.A. Modeling the Effect of Surface Modification of Gold Nanoparticles Irradiated with Co-60 on the Secondary Particles Emission Spectrum. Doklady Physics. 2018. Vol. 63. No. 3. pp. 96-99.

Статья
2018 год

Nadysум G., Tikhomirov A.S., Lin M., Yang Y., Dezhenkova L.G., Chen H., Kaluzhny D.N., Schols D., Shtil A.A., Shchekotikhin A.E., Chueh P.J. Aminomethylation of heliomycin: Preparation and anticancer characterization of the first series of semi-synthetic derivatives. European Journal of Medicinal Chemistry. 2018. Vol. 143. pp. 1553-1562.

Статья
2018 год

Petrova A., Ol'Shevskaya V., Zaitsev A., Tatarskiy V.V., Kalinina E., Andreev Y., Chernov N., Shtil A.A. Antioxidant mechanisms in ovary adenocarcinoma cells resistant to cisplatin do not rescue from photonecrosis: implications for photodynamic therapy. FEBS Open Bio. 2018. Vol. 8. No. S1. pp. 214.

Статья
2018 год

Prilepskii A.Y., Fakhardo A.F., Drozdov A.S., Vinogradov V.V., Dudanov I.P., Shtil A.A., Bel'Tyukov P., Shibeko A., Koltsova E., Nechipurenko D., Vinogradov V.V. Urokinase-conjugated magnetite nanoparticles as a promising drug delivery system for targeted thrombolysis: synthesis and preclinical evaluation. ACS Applied Materials and Interfaces. 2018. Vol. 10. No. 43. pp. 36764-36775.

Статья
2018 год

Zverev V.I., Pyatakov A.P., Shtil A.A., Tishin A.M. Novel applications of magnetic materials and technologies for medicine. Journal of Magnetism and Magnetic Materials. 2018. Vol. 459. pp. 182-186.

Статья
2018 год

Shaikhutdinova N.D., Shaikhutdinov T.F., Frolov G.A., Borisova A.I., Akopdzhanov A.G., Shtil A.A. Design of nanodispersed magnetoactive systems for targeted drug delivery. Nanotechnologies in Russia. 2018. Vol. 13. No. 5-6. pp. 317-321.

Тезисы
2018 год

Высокоэлектроноплотные наноматериалы для онкотераностики

Статья
2018 год

Morozov V.N., Belousov A.V., Krusanov G.A., Kolyvanova M.A., Chernyaev A.P., Shtil A.A. Secondary Electron Spectral Changes of Irradiated Gold Nanoparticle Caused By PEGylation. KnE Energy & Physics. 2018. pp. 278–282.

Статья
2018 год

Pimentel B., Caraballo-Vivas R.J., Checca N.R., Zverev V.I., Salakhova R.T., Makarova L.A., Pyatakov A.P., Perov N.S., Tishin A.M., Shtil A.A., Rossi A.L., Reis M.S. Threshold heating temperature for magnetic hyperthermia: controlling the heat exchange with the blocking temperature of magnetic nanoparticles. Journal of Solid State Chemistry. 2018. Vol. 260. pp. 34-38.

Статья
2018 год

Lukasheva E.V., Kotovshchikov Y.N., Latyshev G.V., Kalinina E.V., Shtil A.A., Kolotova E.S., Lukashev N.V. Transition metals catalyzed reactions–a new approach to the aryl-, azolyl-and triazolylsubstituted steroids–active compounds against human MCF7 breast and SCOV3 ovarian carcinoma cells. FEBS Open Bio. 2018. Vol. 8. No. S1. pp. 238.

Статья
2018 год

Kalinina E.V., Andreev Y.A., Lubova K.I., Petrova A.S., Shtil A.A., Chernov N.N. Redox-dependent change in the expression of genes controlling cellular ROS/antioxidants balance under formation of cancer cell resistance to cisplatin. FEBS Open Bio. 2018. Vol. 8. No. S1. pp. 357.

Статья
2018 год

Antonenko T.A., Shtil A.A., Milaeva E.R. Coordination and Organometallic Compounds with 2,6-di-tert-butylphenol fragments. Synthesis, Structure and Biological Activity. Сборник тезисов всероссийского кластера конференций по неорганической химии "InorgChem2018". 2018. pp. 160.

Статья
2018 год

Belousov A.V., Morozov V.N., Krusanov G.A., Kolyvanova M.A., Chernyaev A.P., Shtil A.A. Spectra of secondary particles generated upon virtual irradiation of gold nanosensitizers: Implications for surface modification. Biomedical Physics and Engineering Express. 2018. Vol. 4. No. 4. pp. 045023.

Тезисы
2017 год

DNA nanomachines for targeting nucleic acids in cancer cells

Тезисы
2017 год

Mechanisms of antioxidant protection and photoinduced death in cisplatin-sensitive and-resistant ovarian adenocarcinoma cells

Статья
2017 год

Kostyukov A.A., Nekipelova T.D., Radchenko A.S., Golovina G.V., Klimovich O.N., Shtil A.A., Codognato D., Goncalves P., Pavanelli A., Ferreira L.P., Amado A.M., Borisevich Y.E., Kuzmin V.A. Triplet states of the complexes of biscarbocyanine dye with albumin. High Energy Chemistry. 2017. Vol. 51. No. 2. pp. 148-150.

Статья
2017 год

Gornostaev L., Tsvetkov V., Markova A., Lavrikova T., Khalyavina Y., Kuznetsova A., Kaluzhny D., Shunayev A., Tsvetkova M., Glazunova V., Chernyshev V., Shtil A.A. The Oxime Derivatives of 1-R-1H-Naphtho[2,3-d][1,2,3]triazole-4,9-dione 2-oxides: Synthesis and Properties. Anti-Cancer Agents in Medicinal Chemistry. 2017. Vol. 17. No. 13. pp. 1814-1823.

Статья
2017 год

Vasilyeva S.V., Shtil A.A., Petrova A.S., Balakhnin S.M., Achigecheva P.Y., Stetsenko D.A., Silnikov V.N. Conjugates of phosphorylated zalcitabine and lamivudine with SiO2 nanoparticles: Synthesis by CuAAC click chemistry and preliminary assessment of anti-HIV and antiproliferative activity. Bioorganic and Medicinal Chemistry. 2017. Vol. 25. No. 5. pp. 1696-1702.

Статья
2017 год

Kostyukov A.A., Pozdnyakova N.V., Shevelev A.B., Radchenko A.S., Golovina G.V., Klimovich O.N., Shtil’ A.A., Codognato D., Goncalves P., Pavanelli A., Ferreira L.P., Amado A.M., Borisevich Y.E., Kuzmin V.A. Complexes of alpha-fetoprotein and serum albumin with biscarbocyanine dye. High Energy Chemistry. 2017. Vol. 51. No. 3. pp. 233-235.

Статья
2017 год

Volkova Y.A., Chernoburova E.I., Petrova A.S., Shtil A.A., Zavarzin I.V. Reactions of hydrazones derived from oxamic acid thiohydrazides. Phosphorus, Sulfur and Silicon and the Related Elements. 2017. Vol. 192. No. 2. pp. 237-240.

Статья
2017 год

Shtil A.A., Miyoshi N., Karaya K., Shimada I., Tanaka H., Sakurai Y., Suzuki M., Zaitsev A.V., Ol’Shevskaya V., Rychkov G., Ono K., Kalinin V. Combination therapy of tumor model with pdt in radiological regions. Journal of International Scientific Publications: Materials, Methods and Technologies (Online). 2017. Vol. 11. pp. 395-402.

Тезисы
2017 год

PEGYLATION MODULATES THE SPECTRUM OF SECOND-ARY ELECTRONS UPON IRRADIATION OF GOLD NANO-PARTICLES: A MONTE-CARLO CALCULATION

Статья
2017 год

Andreeva Y.I., Drozdov A.S., Fakhardo A.F., Cheplagin N.A., Shtil A.A., Vinogradov V.V. The controllable destabilization route for synthesis of low cytotoxic magnetic nanospheres with photonic response. Scientific Reports. 2017. Vol. 7. pp. 11343.

Тезисы
2017 год

Mechanisms of antioxidant protection and photoinduced death in cisplatin-sensitive and-resistant ovarian adenocarcinoma cells

Статья
2017 год

Silva E.R., Pavanelli A.L., Mostaco L.B., Schaberle F.A., Galembeck S.E., Goncalves P.J., Costa E Silva R., Ferreira L.P., Nekipelova T.D., Kostyukov A.A., Radchenko A.S., Shtil A.A., Kuzmin V.A., Borissevitch I.E. Phototransformation of cyanine dye with two chromophores. Effects of oxygen and dye concentration. Journal of Photochemistry and Photobiology A: Chemistry. 2017. Vol. 349. pp. 42-48.

Статья
2017 год

Shtil A.A., Ol'Shevskaya V.A., Zaitsev A.V., Radchenko A.S., Petrova A.S., Markova A.A., Miyoshi N., Borissevitch I.E., Kuzmin V.A. Chemical modifications of tetrapyrrole and carbocyanine scaffolds: On the road to optimized antitumor photosensitizers. Photodiagnosis and Photodynamic Therapy. 2017. Vol. 100. No. 17. pp. A24-A25.

Статья
2016 год

Tishin A.M., Shtil A.A., Pyatakov A.P., Zverev V.I. Developing antitumor magnetic hyperthermia: Principles, materials and devices. Recent Patents on Anti-cancer Drug Discovery. 2016. Vol. 11. No. 4. pp. 360-375.

Повышение квалификации

Повышение квалификации
2023 год
Организация и поддержка образовательного процесса в цифровой образовательной среде

Российская Федерация, Санкт-Петербург

Повышение квалификации
2019 год
Электронная информационно-образовательная среда Университета ИТМО

Российская Федерация, Санкт-Петербург